Substituted DI- and tripeptide inhibitors of protein: farnesyl t

Details Substituted DI- and tripeptide inhibitors of protein: farnesyl t Substituted DI- and tripeptide inhibitors of protein: farnesyl t

1996-06-27

1998-11-03

Tsang, Cecilia J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Peptide containing doai

514 18, 530331, A61K 3805, A61K 3806

Patent

active

058308687

ABSTRACT:
Novel inhibitors of protein:farnesyl transferase enzyme are described, as well as methods for the preparation and pharmaceutical compositions of the same, which are useful in controlling tissue proliferative diseases, including cancer and restenosis.

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