Substituted bicylic thiophene derivatives, compositions...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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Details

C514S443000, C546S114000, C549S050000

Reexamination Certificate

active

10527762

ABSTRACT:
The present invention addresses substituted thiophene derivatives, as well as compositions containing such compounds and methods of treatment. The compounds in the present invention are glucagon antagonists. The compounds block the action of glucagon at its receptor and thereby decrease the levels of plasma glucose providing a treatment of diabetes.

REFERENCES:
Fujita et al. “Synthesis and Bioactivities of Novel Bicylic Thiophenes and 4,5,6,7-Tetrahydrothieno[2,3-c]pyridines as Inhibitors of Tumor Necrosis Factor-a (TNF-a) Production” Bioorganic and Medicinal Chemistry Letters, 2002, vol. 12, pp. 1897-1900.
Fujita, et al—Database Cas Online on STN, Chem. Abstra., Accession No. 2002:510557, 2002.
Fujita, M. et al., “Snthesis and Bioactivities of Novel Bicylic Thiophenes and 4,5,6,7-Tetrahydrothienol[2,3-c]pyridines as Inhibitors of Tumor Necrosis Factor-alpha (TNF-alpha) Production” Bioorganic & Medicinal Chemistry Letters, vol. 12, pp. 1897-1900, 2002.

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