Substituted bicyclocarboxyamide compounds

Details Substituted bicyclocarboxyamide compounds Substituted bicyclocarboxyamide compounds

2011-06-21

2011-06-21

Andres, Janet (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C514S314000, C514S406000, C548S375100

Reexamination Certificate

active

07964732

ABSTRACT:
This invention provides a compound of the formulaThese compounds are useful for the treatment of disease conditions caused by overactivation of the VR1 receptor such as pain, or the like in mammal. This invention also provides a pharmaceutical composition comprising the above compound.

REFERENCES:
patent: 5580983 (1996-12-01), Kraus
patent: 6774136 (2004-08-01), Gerlach et al.
patent: 6979686 (2005-12-01), Naraian et al.
patent: 7084176 (2006-08-01), Morie et al.
patent: 7425641 (2008-09-01), Ries et al.
patent: 2003/0232818 (2003-12-01), Anderson et al.
patent: 2004/0102449 (2004-05-01), Wu et al.
patent: 2005/0009812 (2005-01-01), Seko et al.
patent: 2005/0020644 (2005-01-01), Bisaha et al.
patent: 2005/0165032 (2005-07-01), Norman et al.
patent: 2005/0165046 (2005-07-01), Hulme et al.
patent: 2005/0165049 (2005-07-01), Hulme et al.
patent: 2006/0183909 (2006-08-01), Schmitt et al.
patent: 2007/0105943 (2007-05-01), Nakamoto et al.
patent: 4423353 (1996-01-01), None
patent: 0492178 (1992-07-01), None
patent: 0719760 (1999-09-01), None
patent: 2827599 (2003-01-01), None
patent: 2389580 (2003-12-01), None
patent: WO 9403432 (1994-02-01), None
patent: WO 9509159 (1995-04-01), None
patent: WO 9631475 (1996-10-01), None
patent: WO 9924442 (1999-05-01), None
patent: WO 9926927 (1999-06-01), None
patent: WO 0042026 (2000-07-01), None
patent: WO 0042213 (2000-07-01), None
patent: WO 0064888 (2000-11-01), None
patent: WO 0071512 (2000-11-01), None
patent: WO 0073283 (2000-12-01), None
patent: WO 0076970 (2000-12-01), None
patent: WO 0076971 (2000-12-01), None
patent: WO 0110823 (2001-02-01), None
patent: WO 0147866 (2001-07-01), None
patent: WO 0200651 (2002-01-01), None
patent: WO 0216318 (2002-02-01), None
patent: WO 0234718 (2002-05-01), None
patent: WO 02080928 (2002-10-01), None
patent: WO 02085908 (2002-10-01), None
patent: WO 02100819 (2002-12-01), None
patent: WO 03014064 (2003-02-01), None
patent: WO 03029210 (2003-04-01), None
patent: WO 03030937 (2003-04-01), None
patent: WO 03035621 (2003-05-01), None
patent: WO 03045920 (2003-06-01), None
patent: WO 03068749 (2003-08-01), None
patent: WO 03080578 (2003-10-01), None
patent: WO 03080596 (2003-10-01), None
patent: WO 03086377 (2003-10-01), None
patent: WO 03104178 (2003-12-01), None
patent: WO 2004019933 (2004-03-01), None
patent: WO 2004047743 (2004-06-01), None
patent: WO 2004052370 (2004-06-01), None
patent: WO 2004058164 (2004-07-01), None
patent: WO 2004058176 (2004-07-01), None
patent: WO 2004069792 (2004-08-01), None
patent: WO 2004078114 (2004-09-01), None
patent: WO 2004080463 (2004-09-01), None
patent: WO 2004104018 (2004-12-01), None
patent: WO 2004108133 (2004-12-01), None
patent: WO 2004113331 (2004-12-01), None
patent: WO 2005003084 (2005-01-01), None
patent: WO 2005009962 (2005-02-01), None
patent: WO 2005021509 (2005-03-01), None
patent: WO 2005021553 (2005-03-01), None
patent: WO 2005033079 (2005-04-01), None
patent: WO 2005035526 (2005-04-01), None
patent: WO 2005087742 (2005-09-01), None
patent: WO 2005105760 (2005-11-01), None
patent: WO 2006016548 (2006-02-01), None
Vippagunta et al., Crystalline Solids, 48 Adv. Drug Delivery Rev. 3-26 (2001).
Simon Frantz, The Trouble with Making Combination Drugs, 5 Nature Rev. 881-82 (2006).
Siu, et al., Organic & Biomolecular Chemistry (2005), 3(17). pp. 3140-3160 (XP002478714).
Kariya, et al., Neuroscience Letters, vol. 392, pp. 2132-215 (2006).
Maeda, et al., Biol. Pharm. Bull., vol. 28(5), pp. 649-853 (2005).
Ding, et al., J. Med. Chem. vol. 48, p. 3171-3181 (2005).
Maeda, et al., Biorganic & Medicinal Chemistry, vol. 12, pp. 4351-4360 (2004).
Halder, et al., Science of Synthesis, vol. 16(9), pp. 251-313 (2004).
Uesato, et al., Bioorganic & Medicinal Chemistry Letters. vol. 12, pp. 1347-1349 (2002).
Buolamwini, et al., J. Med. Chem. vol. 45, pp. 841-852 (2002).
Marsilje, et al., Bioorganic & Medicinal Chemistry Letters, vol. 20, pp. 477-481 (2000).
Stanczak, et al., Pharmazie, vol. 53(3), pp. 156-161 (1998).
Burke, et al., J. Med. Chem., vol. 38, pp. 4171-4178 (1995).
Burke, et al., Bioorganic & Medicinal Chemistry Letters, vol. 2(12), pp. 1772-1774 (1992).
Lanza, et al., J. Med. Chem., vol. 35, pp. 252-258 (1992).
El-Kerdawy, et al., J. Pharmaceutical Sciences, vol. 73(11), pp. 1652-1653 (1984).
Nair, et al., J. Org. Chem., vol. 38(12). pp. 2185-2189 (1973).

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