Substituted bicyclic phosphoramides and derivatives thereof

Details Substituted bicyclic phosphoramides and derivatives thereof Substituted bicyclic phosphoramides and derivatives thereof

1994-01-13

1996-08-06

Shah, Mukund J.

Organic compounds -- part of the class 532-570 series

Organic compounds

Four or more ring nitrogens in the bicyclo ring system

546 22, 544337, 548119, 568 12, 558 75, 562507, C07D41314, A61K 3133

Patent

active

055435173

ABSTRACT:
This invention relates to substituted bicyclic phosphoramides and derivatives thereof, useful as retroviral protease inhibitors and as standards and reagents in determining the ability of a potential pharmaceutical to inhibit viral replication or HIV protease, to pharmaceutical compositions comprising such compounds, and to methods of using these compounds for treating viral infection.

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