Substituted an unsubstituted benzooxathiazoles and compounds...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C514S373000, C514S439000, C548S122000, C548S126000, C548S207000, C549S033000

Reexamination Certificate

active

10939936

ABSTRACT:
The invention relates to substituted and unsubstituted 3H-benzo[1,2,3]oxathiazole 2,2-dioxides, 1,3-dihydrobenzo[1,2,5]thiadiazole 2,2-dioxides and 1,3-dihydro-benzo[c]isothiazole 2,2-dioxides, to their preparation and to their use in medicaments.

REFERENCES:
patent: 3539584 (1970-11-01), Judd et al.
patent: 4562185 (1985-12-01), Jager et al.
patent: 5130432 (1992-07-01), Cooper et al.
patent: 5504095 (1996-04-01), Nakane et al.
patent: 5750471 (1998-05-01), Kamireddy et al.
patent: 5789436 (1998-08-01), Kato et al.
patent: 5874382 (1999-02-01), Kamireddy et al.
patent: 6566390 (2003-05-01), Petry et al.
patent: 7-325942 (1995-12-01), None
patent: WO92/05164 (1992-04-01), None
patent: PCT/EP96/03008 (1996-07-01), None
patent: WO98/32438 (1998-07-01), None
patent: WO98/32439 (1998-07-01), None
patent: WO99/11264 (1999-03-01), None
patent: WO99/36069 (1999-07-01), None
patent: WO00/05216 (2000-02-01), None
patent: WO 00/06557 (2000-02-01), None
Tickner et al., An efficient synthesis of catechol cyclic sulfates Synthetic Communications (1994) 24 (11), 1631-1637.
Kingston et al., High yield synthesis of cyclic phosphites, phosphates, sulphites and sulphates of catechol and glycol mediated by hypervalent silicon centres, Tetrahedron Letters, 1997, 38, 27, 4841-4844.
Acheson et al., Acidic epinephrine analogs derived from 1H,3H-2, 1,3-benzothiadazole 2,2-dioxide and from trifluoromethanesulfonanilide. New synthesis of 1H,3H-2, 1,3-benzothiadiazole 2,2-dioxide, J. Med. Chem.; 1981; 24(11); 1300-1304.
Andersen et al., Acidity of Cyclic Sulfamates: Study of Substituted 1,2,3-Benzoxathiazole 2,2-Dioxides and Theoretical Investigation of the Effect of Conformation on Acidity, J. Org. Chem.; 1995; 60(7); 2003-2007.
Chrostowska et al., Application of Photoelectron Spectroscopy to Molecular Properties, 57 UV Photoelectron Spectroscopy Studies of the Products of Thermal Extrusion of Sulfur Dioxide from Benzosultams pp. 313-318, Published Online: Dec. 17, 1999.
Meyer et al., Structure-Activity Studies for a Novel Series of N-(Arylethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-ylmethyl)-N-methylamines Possessing Dual 5-HT Uptake Inhibiting and 2-Antagonistic Activities, J. Med. Chem.; (Article); 1997; 40(7); 1049-1062.
Adcock, W., et. al., Substituent Effects by Fluorine-19 Nuclear Magnetic Resonance: Polar and .pl.-Electron Effects, CA:86:154751 abs of Aust J Chem 29(12) pp. 2571-2581 (1976).
Andersen, K.K., et. al., Acidity of Cyclic Sulfamates: Study of Substituted 1,2,3-Benzoxathiazole 2,2-Dioxides and Theoretical Investigation of the Effect of Conformation on Acidity , CA:123:198187 abs of Journal of Organic Chemistry 60(7) pp. 2003-2007 (1995)*
Andersen, K.K., et al., Reactivity of Nucleophiles Towards X-3-(p-Tolylsulfonyl)1,2,3-Benzoxathiazole 2,2-Dioxides: Kinetics, Activation Volumes and Mechanism, Journal of Physical Organic Chemistry 1997, vol. 10, pp. 175-181.
Anderson, K.K., et al., 1,2,3-Benzoxathiazole 2,2-Dioxide: Synthesis, Mechanism of Hydrolysis, and Reactions with Nucleophiles, CA:115:232139 abs of Journal of Organic Chem 56(23) pp. 6508-6516 (1991).
Bekdemir, et al., CA:136:309895 abs of Journal of Molecualr Struct. 604(2-3) pp. 239-244 (2002).
Grigg, R., et. al., Rhodium Catalyzed [2+2+2]—Cycloadditions of Acetylenes, CA:110:7815 abs of J Chem Soc Perkin Trans 1 (6) pp. 1357-1364 (1988).
Horner, et. al., Additional Ring Opening Reactions of Benzocyclobutene, abs of Justus Liebigs Ann Chem 714 pp. 91-111 (1968).
Ibragimov, M.P., et al., Reactions of 4-Nitro-2-Thiaindan Sulfone, CA:80:82552 abs of Dokl Akad Nauk Tadz SSR 16(10) pp. 27-28 (1973).
Ibragimov, M.P., et. al., Synthesis and Reactions of 4-Nitro-substituted Derivatives of 5,6-Dimethyl-2-Thiaindan Sulfone and Sulfoxide, CA:87:84750 abs of Inst Khim Dushanbe USSR 20(3) pp. 32-33 (1977).
Ibragimov, M.P., et. al., Synthesis of 2-Thioindan and Some of its Derivatives, CA:77:139695 abs of Dokl. Akad. Nauk. Tadz. SSR 15(4) pp. 26-27 (1972).
Kanematsu, K., et. al., One-pot Access to Benzosulfolenes (1,3-Dihydrobenzo [c] Thiophene S,S-Dioxides) Via Allenyl Furfuryl (2-Furylmenthyl) Sulfone Intramolecular Cycloaddition Strategy , CA:117:69687 abs of J Chem Soc Chem Commun. (10) pp. 735-736 (1992).
Lanzetta, P.A., et. al., An improved Assay for Nanomole Amounts of Inorganic Phosphate , Analytical Biochemistry vol. 100, 95-97 (1979).
Levy, L.A., et. al., The Synthesis of 2,3,6,7-Tetrasubstituted Naphthalenes: 2,3,6,7-Tetrachloronaphthalene, CA: 136:309895 abstract of Journal of Molecular Struct, 604(2-3) pp. 239-244 (1983).
N. K. Tonks et al., Characterization of the Major Protein-tyrosine phosphatases of Human Placenta, Journal of Biological Chemistry, vol. 263, No. 14, May 15, 1988, pp. 6731-6737.
Nasyrov, I.M., et. al., Halogenation of 2-Thiaindan 2,2-Dioxide, CA:84:89930 abs of Khim Tadzh. Editor Solozhenkin (1973) pp. 107-110.
Nasyrov, I.M., et. al., Synthesis and Oxidation of 5,6-Dimethyl-2 Thiaindan, CA:82:43118 abs of Dokl Akad Nauk Tadz, SSR 17(6) pp. 28-29 (1974).
Oppolzer, W., et. al., The enantioselective synthesis of (+)-Estradiol from 1,3-Dihydrobenzo (c) Thiophene-2,2-dioxide by Successive Thermal Sulfur Dioxide Extrusion and Cycloaddition Reactions. Preliminary Communication, CA:94:121179 abs of Helv Chim Acta 63(6) pp. 1703-1705 (1980).
Summer, M.D., et. al., A Manual of Methods for Baculovirus Vectors and Insect Cell Procedures , Department of Entomology Texas Agricultural Experiment Station and Texas A & M University, Bulletin No. 1555, May 1987.
T.R. Burke et al., Small Molecule Interactions with Protein-Tyrosine Phosphatase PTP1B and Their Use in Inhibitor Design, Biochemistry, vol. 35, 1996, pp. 15989-15996.
Tyle, Praveen, Iontophoretic Devices for Drug Delivery, Pharmaceutical Research, vol. 3, No. 6, 1986 pp. 318-326.
W. Cromlish et al., Selective Inhibition of Cyclooxygenase-1 and -2 Using Intact Insect Cell Assays, Biochemical Pharmacology, vol. 52, 1996, pp. 1777-1785.
1,3-Dihydro-2,1-Benzisothiazole 2,2-Dioxide, Beilstein Institut zur Forderung der Chyemischen Wissenschaften, Frankfurt am Main, DE; retrieved from Beilstein Xfire Accession No. 4387065, Zusammenfassung, Zusammenfassung, Journal of Heterocyclic Chemistry, Nr. 23, 1986 Seiten 1645-1649.
1,3-dihydro-Benzo(c)Thiophene-2,2-Dioxide, Beilstein Institut zur Forderung der Chyemischen Wissenschaften, Frankfurt am Main, DE; retrieved from Beilstein Xfire Accession No. 117793, Journal of American Chemical Soc., Nr. 81 (1959) Seiten 4266.
1,3-dihydro-Benzol[1,2,5]Thiadiazole-2,2-Dioxide, Beilstein Institut zur Forderung der Chyemischen Wissenschaften, Frankfurt am Main, DE; retrieved from Beilstein Xfire Accession No. 608462, Zusammenfassung, Journal of American Chemical Soc. C. (1971) Seiten 993-999.
3H-1,2,3-Benzoxathiazole-2,2-Dioxide, Beilstein Institut zur Forderung der Chyemischen Wissenschaften, Frankfurt am Main, DE; retrieved from Beilstein Xfire Accession No. 4800778, Zusammenfassung, Journal of Organic Chemistry, Bd. 56, Nr. 23, 1991 Seiten 6508-6516.
3H-Benzo[d][1,2]Oxathiol-2,2-Dioxide, Beilstein Institut zur Forderung der Chyemischen Wissenschaften, Frankfurt am Main, DE; retrieved from Beilstein Xfire Accession No. 4407, Chemische Berichte, Nr. 31, (1898) Seite 1857.
Benzo[1,3,2]Dioxathiol-2,2-Dioxide, Beilstein Institut zur Forderung der Chyemischen Wissenschaften, Frankfurt am Main, DE; retrieved from Beilstein Xfire Accession No. 2047037, Zusammenfassung, C.R. Herd, Seances Acad Sci. Nr. 203, (1936) Seite 194.

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