Substituted aminothienopyridines, pharmaceutical composition and

Details Substituted aminothienopyridines, pharmaceutical composition and Substituted aminothienopyridines, pharmaceutical composition and

1997-01-08

1999-01-05

Rotman, Alan L.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

546114, C07D47104, C07D48704, A61K 3144

Patent

active

058563350

ABSTRACT:
This application relates to compounds of the formula ##STR1## wherein R.sup.1, R.sup.2, R.sup.3, m and n are as defined in the specification which are useful as modulators of neurotransmitter function such as serotonergic and adrenergic, and as such are useful as antidepressants, anxiolytics, atypical antipsychotics, antiemetics, and for the treatment of personality disorders such as obsessive compulsive disorders. Certain of the compounds are also useful as glycine partial agonists.

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