Substituted 8-phenylisoxazolo[4,3-e][1,4]diazepin-5-ones

Details Substituted 8-phenylisoxazolo[4,3-e][1,4]diazepin-5-ones Substituted 8-phenylisoxazolo[4,3-e][1,4]diazepin-5-ones

1984-05-31

1985-04-30

Bond, Robert T.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

2602393B, 548245, A61K 3155, C07D49804, C07D26114

Patent

active

045144109

ABSTRACT:
This invention relates to substituted 8-phenylisoxazolo[4,3-e][1,4]diazepin-5-ones of the formula ##STR1## wherein R is lower alkyl; R.sub.1 is hydrogen, amino alkyl, propargyl and lower alkyl; X is oxygen and sulfur; and Y is halogen, trifluoromethyl, lower alkyl, lower alkoxy and hydrogen. The compounds of this invention display useful anxiolytic and anticonvulsant activites.

REFERENCES:
patent: 4172079 (1979-10-01), Love
Dal Piaz et al., "Synthesis", pp. 664-665, (Oct. 1975), Communications.
Jaunin, "Helv. Chim. Acta", (1974), vol. 57 (7), pp. 1934-1942.
Otsuji et al., "Bull. Chem. Soc. Japan", vol. 44, pp. 223-226 (1971).

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