Substituted 5-aryl-benzothiepines having activity as inhibitors

Details Substituted 5-aryl-benzothiepines having activity as inhibitors Substituted 5-aryl-benzothiepines having activity as inhibitors

1999-03-24

2000-08-22

Lambkin, Deborah C.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

514431, 514249, 514314, 544236, 544176, C07D33700, C07D48700, A61K 3138, A61K 31495

Patent

active

061074942

ABSTRACT:
Provided are novel benzothiepines, derivatives, and analogs thereof; pharmaceutical compositions containing them; and methods of using these compounds and compositions in medicine, particularly in the prophylaxis and treatment of hyperlipidemic conditions such as those associated with atherosclerosis or hypercholesterolemia, in mammals.

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