Substituted 1-propiolylpiperazine compounds, their...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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Details

C514S253100, C514S254020, C514S254030, C544S363000, C544S364000, C544S367000, C544S369000

Reexamination Certificate

active

11649156

ABSTRACT:
Substituted 1-propiolylpiperazine compounds corresponding to formula Iin which X denotes N or C—R2, and n is an integer from 0 to 8, a method for producing such substituted 1-propiolylpiperazine compounds, pharmaceutical compositions containing such substituted 1-propiolylpiperazine compounds, and the use of such substituted 1-propiolylpiperazine compounds for modulating mGluR5 receptor activity or for treating or inhibiting pain and various other conditions, especially conditions at least partly mediated by the mGluR5 receptor.

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patent: WO 2004/029044 (2004-04-01), None
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