Substituted 1,4-diazapine caprolactams useful for treatment of H

Details Substituted 1,4-diazapine caprolactams useful for treatment of H Substituted 1,4-diazapine caprolactams useful for treatment of H

1993-03-30

1997-09-02

Shah, Mukund J.

Organic compounds -- part of the class 532-570 series

Organic compounds

Unsubstituted hydrocarbyl chain between the ring and the -c-...

540484, 540485, C07D24308, A61K 3155

Patent

active

056633335

ABSTRACT:
This invention relates to novel substituted caprolactams, including 4-azacaprolactams, and derivatives thereof which inhibit HIV protease and are useful for treatment of HIV disease. Also included in this invention are pharmaceutical compositions containing such caprolactams, and to methods of using such caprolactams for the treatment of HIV disease.

REFERENCES:
patent: 4002612 (1977-01-01), Schwan
patent: 4096140 (1978-06-01), Simpson
patent: 4466916 (1984-08-01), Lai et al.
Tetrahedron vol. 49, No. 8, pp. 1547-1556, 1993.
Kimura, Agric. Biol. Chem. (1989) 53: 1811.

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