Structure-based modulators of B1 G-protein coupled receptors

Data processing: measuring – calibrating – or testing – Measurement system in a specific environment – Biological or biochemical

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C703S011000

Reexamination Certificate

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07869958

ABSTRACT:
The present invention relates to a method for identifying modulators of B1 G-protein coupled receptors. The present invention also relates to a method for identifying an antagonist or agonist of the corticotropin-releasing factor receptor 2 (CRFR2). The present invention also relates to a method for improving antagonists or agonists of CRFR2. The present invention also relates to the three-dimensional structure of CRFR2 as representative of the B1 GPCR subfamily and its use as a basis for rational drug design of antagonist or agonists of B1 GPCRs.

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