Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Cyclopentanohydrophenanthrene ring system doai
Patent
1997-07-18
1999-03-09
Dees, Jose G.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Cyclopentanohydrophenanthrene ring system doai
514182, 552522, 552611, A61K 3156, C07J 300, C07J 4100
Patent
active
058801154
ABSTRACT:
Sulfatase inhibitor compounds having the formula: ##STR1## wherein X, Y, R.sub.1, R.sub.2 and R.sub.3 are as defined in the specification. The compounds are useful in the treatment of estrogen dependent illnesses. Methods for synthesizing these compounds are also disclosed.
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Li Pui-Kai
Selcer Kyle W.
Badio Barbara
Dees Jos,e G.
Duquesne University of the Holy Ghost
Meyers Diane R.
Silverman Arnold B.
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