Stereospecific synthesis of 2(R)-2-methyl-3-dimethylamino-propio

Organic compounds -- part of the class 532-570 series – Organic compounds – Amino nitrogen containing

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564342, C07C20946, C07C20968

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051324571

ABSTRACT:
In a method for producing 2(R)-2-methyl-3-dimethylamino-propiophenone (d-DAMP), a chiral ester of the formula ##STR1## wherein R is an alkyl of from 1 to about 5 carbon atoms, is provided. The chiral easter of formula (I) is converted into a chiral amino-alcohol of the formula ##STR2## and the chiral amino-alcohol is oxidized so as to form d-DAMP.

REFERENCES:
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