Stereoselective process for the production of dioxolane...

Chemistry: molecular biology and microbiology – Process of utilizing an enzyme or micro-organism to destroy... – Resolution of optical isomers or purification of organic...

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

C435S118000, C435S135000, C435S088000, C435S019000, C514S04400A

Reexamination Certificate

active

07955835

ABSTRACT:
The present invention relates to a process for producing compounds of formula (I) and (VII); said process comprising the steps of: a) subjecting a compound of formula (II) to an enzymatic diastereomeric resolution in the presence of a suitable amount of enzyme chosen from Pig Liver Esterase or Porcine Pancreatic Lipase b) recovering said compounds of formula (I) and (VII). The invention also provides a process for producing compounds of formula (III) and (X); said process comprising the steps of: a) subjecting a compound of formula (IV) to an enzymatic diastereomeric resolution in the presence of a suitable amount of enzyme chosen fromCandida Antarctica“A” lipase,Candida Antarctica“B” lipase,Candida LypoliticaLipase orRhizomucor MieheiLipase b) recovering said compound of formula (III) and (X).

REFERENCES:
patent: 2001/0049372 (2001-12-01), Nguyen-Ba
patent: WO 0039143 (2000-07-01), None
patent: WO 00/47759 (2000-08-01), None
patent: WO 0047759 (2000-08-01), None
Ferrero et al., Monatshefte für Chemie, 2000, vol. 131, p. 585-616.
Adler et al., JBC, 1961, vol. 236, No. 12, p. 3240-3245.
Martinelle et al., Biochimica et Biophysica Acta, 1995, vol. 1258 p. 272-276.
Janes et al: “Protease -Mediated Separation of Cis and Trans Diastereomers of 2(R,S)- benzyloxymethy1-4(S)-carboxylic Acid 1,3-Dioxolane Methy Ester: Intermediates for the Synthesis of Dioxolane Nucleosides” Journal of Organic Chemistry, American Chemical Society, Easton, US, vol. 64, Nov. 19, 1999, pp. 9019-9029, XP002137411.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Stereoselective process for the production of dioxolane... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Stereoselective process for the production of dioxolane..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Stereoselective process for the production of dioxolane... will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-2681310

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.