Stereoselective preparation of substituted piperidines

Details Stereoselective preparation of substituted piperidines Stereoselective preparation of substituted piperidines

1993-09-20

1997-11-11

Reamer, James H.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D21132

Patent

active

056866151

ABSTRACT:
Novel processes are disclosed for the stereoselective preparation of substituted piperidine derivatives of the formulae ##STR1## wherein R.sup.1 and R.sup.2 are defined as below, useful as substance P receptor antagonists and in treating diseases mediated by an excess of substance P.

REFERENCES:
patent: 2355659 (1944-08-01), Nutley et al.
patent: 4267318 (1981-05-01), Hershenson
H. Rodd. Rodd's Chemistry of Carbon Compounds, Elsevier Scientific Publishing Co., pp. 212-213 (1976).
H. House, Modern Synthetic Reactions, Second Edition, W. A. Benjamin, Inc., pp. 3-15 (1972).
Solomons, T W Graham Organic Chemistry (1988) pp. 259-264.

Affiliated with

Also associated with

Rating

Stereoselective preparation of substituted piperidines does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Stereoselective preparation of substituted piperidines, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Stereoselective preparation of substituted piperidines will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-1230466