Stable, high dose, high bulk density ibuprofen granulations for

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Radical -xh acid – or anhydride – acid halide or salt thereof...

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514770, 514781, A61K 916, A61K 934

Patent

active

046096752

ABSTRACT:
Dry granulate pharmaceutical compositions containing 85 to 99 percent by weight of ibuprofen and 1 to 15 percent, by weight of Croscarmellose sodium, types A and/or B (cross-linked sodium carboxymethylcellose) are useful for making ibuprofen compressed tablet and filled capsule formulations containing from about 100 to about 1200 mg. of ibuprofen per dosage unit. They are particularly helpful for making compressed tablets containing from 800 to 1200 mg. of ibuprofen per tablet, which have bioavailability rates similar to those of presently known lower dosage strength ibuprofen tablets.

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patent: 4361580 (1982-11-01), Peck et al.
patent: 4404371 (1983-09-01), Bellmann et al.
patent: 4439453 (1984-03-01), Vogel
patent: 4521594 (1985-06-01), Kanematu
A group of Derwent Abstract card copies, on numbered pp. 2 to 20, disclosing drug formulations, some with Ibuprofen.
Third Supplement to USP XX and to NF XV (1982) pp. 367-368.
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Mallinckrodt brochure (2 pages) for 90% Acetaminophen/10% Starch COMPAP Product.

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