Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Nitrogen containing other than solely as a nitrogen in an...
Reexamination Certificate
2011-08-02
2011-08-02
Wilson, James O (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Nitrogen containing other than solely as a nitrogen in an...
C544S336000, C546S329000, C548S375100, C549S074000, C549S491000, C549S505000, C564S086000
Reexamination Certificate
active
07989497
ABSTRACT:
The present invention relates to compounds of formula (I)wherein X, R1, R2, R3, R4and R5are as defined herein, which are useful for treating diseases which respond to CXCR2 receptor mediators. Pharmaceutical compositions that contain the compounds and processes for preparing the compounds are also described.
REFERENCES:
patent: 6166050 (2000-12-01), Lombardo et al.
patent: 7132445 (2006-11-01), Taveras et al.
patent: 2004/0106794 (2004-06-01), Taveras et al.
patent: 2004/0147559 (2004-07-01), Taveras et al.
patent: 2008/0200523 (2008-08-01), Murthi et al.
patent: 102005035742 (2007-02-01), None
patent: 1818325 (2010-02-01), None
patent: 02/057230 (2002-07-01), None
patent: 02/079122 (2002-10-01), None
patent: 02/083624 (2002-10-01), None
patent: 03/080053 (2003-10-01), None
patent: 2004/011418 (2004-02-01), None
patent: 2005/075447 (2005-08-01), None
patent: 2006/072354 (2006-07-01), None
patent: 2006/084661 (2006-08-01), None
patent: 2006/088920 (2006-08-01), None
patent: 2008/005570 (2008-01-01), None
patent: 2009/005801 (2009-01-01), None
patent: 2009/005802 (2009-01-01), None
patent: 2009/012375 (2009-01-01), None
patent: 2009/073683 (2009-06-01), None
patent: 2010/683802 (2010-06-01), None
patent: 2010/091543 (2010-08-01), None
Yun Feng Xie et al., “Structure-activity relationships of novel, highly potent, selective, and orally active CCR1 antogonists,” Bioorganic & Medicinal Chemistry Letters 15:3367-3372 (Apr. 5, 2007).
Baettig Urs
D'Souza Anne-Marie
Hunt Peter
Press Neil John
Watson Simon James
Devlin Theresa A.
Milstead Mark
Novartis AG
Willis Douglas M
Wilson James O
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