Spiropiperidine derivatives as NK3 antagonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C544S071000

Reexamination Certificate

active

07470684

ABSTRACT:
The present invention relates to a compound of formula Iwherein R1, R2, R3, R4, R7, m and n are as defined herein. These compounds are high potential NK-3 receptor antagonists useful for the treatment of depression, pain, psychosis, Parkinson's disease, schizophrenia, anxiety and attention deficit hyperactivity disorder (ADHD).

REFERENCES:
patent: WO 02/092604 (2002-11-01), None
patent: WO 2005/092858 (2005-10-01), None
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