Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1997-12-04
2000-01-11
Shah, Mukund J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
5142265, 514258, 514373, 514409, 544 6, 544230, 546 17, 546 18, 548207, 548409, 548410, A61K 3144, C07D40102
Patent
active
060136529
ABSTRACT:
Disclosed are spiro-substituted azacycles of formula I are tachykinin receptor antagonists useful in the treatment of inflammatory diseases, pain or migraine, and asthma. In particular compounds of formula I are shown to be neurokinin antagonists.
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Chiang Yuan-Ching P.
Dunn Patrick T.
Koyama Hiroo
Maccoss Malcolm
Mills Sander G.
Billups Richard C.
Coleman Brenda
Merck & Co. , Inc.
Rose David L.
Shah Mukund J.
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