Solid phase synthesis method

Details Solid phase synthesis method Solid phase synthesis method

1998-07-02

1999-08-24

Huang, Evelyn Mei

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D31728

Patent

active

059426322

ABSTRACT:
A solid phase synthesis method and intermediates useful in the process are disclosed for the preparation of diamino diol and diamino alcohol inhibitors of HIV protease.

REFERENCES:
patent: 4506085 (1985-03-01), Yamada
patent: 4808729 (1989-02-01), Deason
Journal of Medicinal Chemistry, 1995, vol. 38, No. 9, "Expedient Method for the Solid-Phase Synthesis of Aspartic Acid Protease Inhibitors Directed toward the Generation of Libraries" by Ellen K. Kick and Jonathan A. Ellman, 1427-1430.
Tet Lett, 1994, vol. 35, "Straightforward and General Method for Coupling Alcohols to Solid Supports", by Lorin A. Thompson and Jonathan A. Ellman, 9333-9336.
Green TW & Wuts PGM. Protective Groups in Organic Synthesis. Second edition. John Wiley & Sons, INC. New York, pp. 224. 225, 231, 248 (1991).

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