Small molecule inhibitors of botulinum neurotoxins

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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Details

C514S438000, C514S461000, C549S029000

Reexamination Certificate

active

07825154

ABSTRACT:
Disclosed herein are methods of inhibiting the activity of Botulinum neurotoxin A metalloprotease with the compounds disclosed herein. Also disclosed are methods of treating, inhibiting or preventing intoxication caused by bacteria of at least one bacterial strain in a subject, and pharmaceutical and cosmetic compositions comprising the compounds disclosed herein.

REFERENCES:
patent: 2005/0251345 (2005-11-01), Bavari et al.
Weidner-Wells et al. “Amidono Benimidazole Inhibitors of Bacerial Two-Component Systems” Bioorganic & Medicinal Chemistry Letters, 2001, vol. 11, pp. 1545-1548.
Mota-Meira et al. “MICs of Mutacin B-Ny266, Nisin A, Vancomycin, and Oxacillin against Bacterial Pathogens” Antimicrobial abents and chemotherapy, Jan. 2000, pp. 24-29.
Anne, J. et al. (1980) “Antifungal and Antibacterial Activities of Diarylamidine Derivatives” Antimicrobial Agents & Chemotherapy 18(2):231-239.
De. Clercq et al. (1980) “Diary1 Amidine Derivatives as Oncornaviral DNA Polymerase Inhibitors” J. Med. Chem. 23:787-795.
Tidwell et al. (1978) “Diarylamidine Derivatives with One or Both of the Aryl Moieties Consisting of an Indole or Indole-like Ring, Inhibitors of Arginine-Specific Esteroproteases” J. Med. Chem. 21(7):613-623.

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