Site-specific inhibitors of histone methyltransferase...

Details Site-specific inhibitors of histone methyltransferase... Site-specific inhibitors of histone methyltransferase...

2011-08-23

2011-08-23

Sullivan, Daniel (Department: 1621)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Radical -xh acid, or anhydride, acid halide or salt thereof...

C514S529000, C560S059000

Reexamination Certificate

active

08003698

ABSTRACT:
The present invention relates to compounds of structural formula I as site-specific inhibitors of histone methyltransferase, where R1and R1is —OCH3or —OH, R2and R2is —OH or —OAc; a process of isolating compound of structural formula Ia, where R1and R1is —OCH3, R2and R2is —OH; a process of preparation of compound of structural formula Ib, where R1and R1is —OCH3, R2and R2is —OAc; a process of preparation of compound of structural formula Ic, where R1and R1is —OH, R2and R2is —OH; and use of compounds of structural formula I for manufacture of a medicament for management of cancer and/or disease conditions in a subject in need thereof.

REFERENCES:
patent: 2002/0197341 (2002-12-01), Lansky
patent: 2004/189599 (2004-07-01), None
patent: 2005/089304 (2005-04-01), None
patent: WO 01/37848 (2001-05-01), None
patent: WO 03/101751 (2003-12-01), None

Affiliated with

Also associated with

Rating

Site-specific inhibitors of histone methyltransferase... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Site-specific inhibitors of histone methyltransferase..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Site-specific inhibitors of histone methyltransferase... will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-2761635