Selective antagonists of A2A adenosine receptors

Details Selective antagonists of A2A adenosine receptors Selective antagonists of A2A adenosine receptors

2007-05-15

2007-05-15

Berch, Mark L. (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Phosphorus containing other than solely as part of an...

C514S234200, C514S228500, C514S263200, C514S263210, C514S263220, C514S263230, C514S263370, C514S263400, C544S061000, C544S118000, C544S244000, C544S276000, C544S277000

Reexamination Certificate

active

11097251

ABSTRACT:
Selective antagonists of A2Aadenosine receptors like those of formula I are provided, wherein Y forms a ring.The novel A2Ablockers are useful for the treatment of Parkinsons disease and other diseases.

REFERENCES:
patent: 4293690 (1981-10-01), Sawa et al.
patent: 4341769 (1982-07-01), Marumoto et al.
patent: 5189027 (1993-02-01), Miyashita et al.
patent: 5681941 (1997-10-01), Cook et al.
patent: 6329381 (2001-12-01), Kurimoto et al.
patent: 6387889 (2002-05-01), Endo et al.
patent: 2004/0043388 (2004-03-01), Come et al.
patent: 2005/0187228 (2005-08-01), Haesslein
Cesnek et al., Collection of Czechoslovak Chemical Communications 68(11), 2201-2218.
Camaioni et al., Bioorganic & Medicinal Chemistry, vol. 6(5) May 1998, pp. 523-533.
Ying Zhao et at., J. Am. Chem., Soc.; 2003; 125(9) pp. 2480-2488.
Klotz, Naunyn-Schmiedeberg's Archives of Pharmacology 367(3) 629-634 (2003).
Baker, J. Org Chem., 19(11) 1793 (1954).
Abiru, J. Med. Chem 35, 2253 (1992).
Gray, Tetrahedron Letters vol. 38, Issue 7, Feb. 17, 1997, pp. 1161-1164.

Affiliated with

Also associated with

Rating

Selective antagonists of A2A adenosine receptors does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Selective antagonists of A2A adenosine receptors, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Selective antagonists of A2A adenosine receptors will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-3747439