Selective acylation of secondary hydroxyl groups

Details Selective acylation of secondary hydroxyl groups Selective acylation of secondary hydroxyl groups

2007-02-13

2007-02-13

Seaman, Margaret D. (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C549S511000

Reexamination Certificate

active

10510063

ABSTRACT:
The invention provides methods and compositions for selectively acylating a specific hydroxyl group in a molecule of interest containing at least two unprotected secondary hydroxyl groups. Although the methods and compositions of the invention have general applicability, they are particularly useful in the selective acylation of taxane molecules.

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