Saccharopeptides and derivatives thereof

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai

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514 18, 514 19, 514 23, 530322, 536 111, 536 53, 536 55, 536 552, A61K 3804, A61K 3170

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058497099

ABSTRACT:
Saccharopeptides and methods of using the novel saccharopeptides are described having the following structural formula I:
wherein W is independently one or more saccharide(s); Y is independently --CO--NH-- or --NH--CO--; and m is an integer greater than or equal to one; or structural formula II:
wherein W is independently one or more saccharide(s); S is a difunctional or polyfunctional alkyl, aryl or aralkyl group, lipid, amino acid or peptide capable of covalently joining together said saccharides; Y is independently --CO--NH-- or --NH--CO--; and n is an integer greater than or equal to zero; or formula III:

REFERENCES:
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