Saccharin derivatives useful as proteolytic enzyme inhibitors an

Details Saccharin derivatives useful as proteolytic enzyme inhibitors an Saccharin derivatives useful as proteolytic enzyme inhibitors an

1994-07-05

1997-07-22

Richter, Johann

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

548210, 544135, 546198, 5462711, 514321, 514338, 5142338, A61K 31535, A61K 31425, C07D41712, C07D41706

Patent

active

056504225

ABSTRACT:
Novel 2-substituted saccharins which inhibit the enzymatic activity of proteolytic enzymes, are useful in the treatment of degenerative diseases and have the formula ##STR1## wherein: L is --O--, --S--, --SO-- or --SO.sub.2 --;

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