Renin inhibitors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Silicon containing doai

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514 64, 514 2, 549 4, 549213, 518110, 518405, 564 8, 558288, 558289, 546 13, 562 7, A61K 3169, A61K 31698, C07D33358

Patent

active

051698412

ABSTRACT:
The invention relates to compounds of the formula 1 ##STR1## in which A.sup.1 denotes a radical of the formulae ##STR2## A.sup.2 is absent or represents a radical of the formula ##STR3## R.sup.2, R.sup.3 and R.sup.4 are as defined in the specification, and X and Y, independently of one another, represent --O-- or --NR.sup.13 --, and to the salts thereof. Also described is a process for the preparation of the compounds of the formula 1, corresponding pharmaceutical products, and the use thereof as medicines, and intermediates for the preparation of these compounds.

REFERENCES:
patent: 4499082 (1985-02-01), Shenvi et al.
Smith, et al., "Principles of Biochemistry: Mammalian Biochemistry," 7th ed., pp. 158-163, McGraw-Hill Book Co., New York (1983).
Hui et al., J. Med. Chem., vol. 30, pp. 1287-1295 (1987).
J. Med. Chem., 1985, vol. 28, pp. 1917-1925, American Chem. Soc., D. H. Kinder et al., "Acylamino Boronic Acids and Difluoroborane . . .".

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