Drug – bio-affecting and body treating compositions – Preparations characterized by special physical form – Tablets – lozenges – or pills
Patent
1996-02-09
1998-06-09
Page, Thurman K.
Drug, bio-affecting and body treating compositions
Preparations characterized by special physical form
Tablets, lozenges, or pills
424465, 424468, 424489, A61K 920, A61K 922
Patent
active
057629617
ABSTRACT:
The invention provides methods of making rapidly soluble tablets of decreased weight compared to similar solid tablets. The invention further provides novel, rapidly soluble tablets of decreased weight compared to similar solid tablets. The tablets offer increased rates of dissolution and disintegration.
REFERENCES:
patent: 3557717 (1971-01-01), Chivers
patent: 3619294 (1971-11-01), Black et al.
patent: 3632357 (1972-01-01), Childs
patent: 3655442 (1972-04-01), Schwer et al.
patent: 4127502 (1978-11-01), Li Mutti et al.
patent: 4158544 (1979-06-01), Louderback
patent: 4327076 (1982-04-01), Puglia et al.
patent: 4327077 (1982-04-01), Puglia et al.
patent: 4588744 (1986-05-01), McHugh
patent: 4678812 (1987-07-01), Bollin, Jr. et al.
patent: 4701417 (1987-10-01), Portenhauser et al.
patent: 4762857 (1988-08-01), Bollin, Jr. et al.
patent: 4865871 (1989-09-01), Livesey et al.
patent: 4883762 (1989-11-01), Hoskins
patent: 4891319 (1990-01-01), Roser
patent: 5026566 (1991-06-01), Roser
patent: 5112616 (1992-05-01), McCarty
patent: 5149653 (1992-09-01), Roser
patent: 5290765 (1994-03-01), Wettlaufer et al.
patent: 5306506 (1994-04-01), Zema et al.
patent: 5348852 (1994-09-01), Bonderman
patent: 5422384 (1995-06-01), Samuels et al.
patent: 5425951 (1995-06-01), Goodrich, Jr. et al.
patent: 5466470 (1995-11-01), Lajoie
patent: 5482720 (1996-01-01), Murphy et al.
patent: 5501861 (1996-03-01), Makino et al.
patent: 5512547 (1996-04-01), Johnson et al.
patent: 5589167 (1996-12-01), Cleland et al.
Dialog.RTM. English Abstract of JP 58-216695 (Dec. 16, 1983).
Dialog.RTM. WPI File 351 Abstract of PCT WO 87/05300 (Sep. 11, 1987).
Sakurai, Y (ed.), "Food General Dictionary" Sixth Edition (The English translation is 10 pages total.).
Kanna et al., "Denaturation of Fish Muscle Protein by Dehydration-V." Bull. Tokai Reg. Fish. Res. Lab. (1974) 77:1-14.
Reasons for Opposition, (1995) 5 pages total.
Supplement of Reasons for Opposition (Dec. 31, 1995), 23 pages total.
Grounds for Rejection, (1995) 6 pages total.
Handbook of Natural Materials for Food Processing, Ninth Edition (Translation to be disclosed at a later date).
Chemical Dictionary, 7.sup.th Edition (Translation to be disclosed at a later date).
Stability and characterization of protein and peptide drugs, Wang et al. (eds.), 1993, table of contents enclosed herewith.
Pogany et al., "A new approach to the theory of tabletting" Acta Pharm. Hung. (1988) 58:49-55.
Doelker, "Recent advances in tableting science" Boll. Chim. Farm. (1988) 127:37-49.
Hiestand et al., "Physical processes of tableting" J. Pharm. Sci. (1977) 66:510-519.
Cooper et al., "Tableting research and technology" J. Pharm. Sci. (1972) 61:1511-1555.
Rudnic et al., "Oral solid doseage forms" Chapter 92, Remington: The Science and Practice of Pharmacy, Nineteenth Edition, Gennaro Ed. (1995) Mack Publishing Company, Pennsylvania vol. II, pp. 1615-1649.
Niwa et al., "Preparation of agglomerated crystals for direct tabletting and microencapsulation by the spherical crystallization technique with a continuous system" Pharm. Res. (1994) 11:478-484.
Franz et al., "Cost evaluation of alternative pharmaceutical tableting processes by simulation" J. Pharm. Sci. (1980) 69:621-628.
Lipps et al., "Characterization of wet granulation process parameters using response surface methodology. 1. Top-spray fluidized bed" J. Pharm. Sci. (1994) 83:937-947.
Drissi-Alami et al., "The effects of the tabletting machine speed on physical characteristics of pharmaceutical powers" J. Pharm. Belg. (1993) 48:43-52.
Ishino et al., "Influence of tabletting speed on compactibility and compressibility of two direct compressible powders under high speed compression" Chem. Pharm. Bull. (1990) 38:1987-1992.
Sendall et al., "A study of powder adhesion to metal surfaces during compression of effervescent pharmaceutical tablets" J. Pharm. Pharmacol. (1986) 38:489-493.
Jetzer, "Measurement of hardness and strength of tablets and their relation to compaction performance of powders" J. Pharm. Pharmacol. (1986) 38:254-258.
Reading et al., "The effects of binder film characteristics on granule and tablet properties" J. Pharm. Pharmacol. (198) 36:421-426.
Paronen et al., "Compressional characteristics of four starches" J. Pharm. Pharmacol. (1983) 35:627-635.
Nakagawa, "Effects of tableting procedures on the preferred orientation of crystalline particles" Chem. Pharm. Bull. (1982) 30:1401-1407.
Elsabbagh et al., "Physical properties and dissolution profiles of acetaminophen and acetylsalicyclic acid tables made from sucrosebased vehicles" Pharmazie (1981) 36:488-492.
Naito et al., "Prediction of tableting problems such as capping and sticking: Theoretical calculations" J. Pharm. Sci. (1977) 66:254-259.
Healey et al., "The mechanical properties of some binders used in tableting" J. Pharm. Pharmac. (1974) 26 Suppl:41P-46P.
York et al., "The effect of temperature on the mechanical properties of some pharmaceutical powders in relation to tableting" J. Pharm. Pharmac. (1972) 24 Suppl:47P-56P.
Sebhatu et al. "Effect of moisture sorption on tabletting characteristics of spray dried (15% amorphous) lactose" Pharm. Res. (1994) 11:1233-1238.
Vromans et al., "Studies on tabletting properties of lactose. Part 1. The effect of intial particle size on binding properties and dehydration characteristics of lactose" Acta Pharm. Suec. (1985) 22:163-172.
Vromans et al., "Studies on tableting properties of lactose. Part 2. Consolidation and compaction of different types of crystalline lactose"
De Boer et al., "Studies on tableting properties of lactose. Part III. The consolidation behaviour of sieve fractions of crystalline .alpha.-lactose
Van Kamp et al., "Studies on tableting properties of lactose. V. Effects of both lubrication and addition of disintegrants on properties of tablets prepared from different types of crystalline lactose" Acta Pharm. Suec. (1986) 23:217-230.
Vromans et al., "Studies on tableting properties of lactose. VI. Consolidation and compaction of spray dried amorphous lactose" Acta Pharm. Suec. (1986) 23:231-240.
Georgakopoulos et al., "The effects of using different grades of PVP and gelatin as binders in the fluidized bed granulation and tableting of lactose" Pharmazie (1983) 38:240-243.
York et al., "Science Papers. The tensile strength and compression behaviour of lactose, four fatty acids, and their mixtures in relation to tableting" J. Pharm. Pharmac. (1973) 25:Suppl:1P-11P.
Blakely et al., "Dry instant blood typing plate for bedside use" Lancet (1990) 336:854-855.
Roser, "Trehalose, a new approach to premium dried foods" Trends in Food Sci. and Tech. (Jul. 1991) pp. 166-169.
Colaco et al., "Trehalose stabilisation of biological molecules" Biotechnol. Internat. (1992) pp. 345-350.
Roser, "Trehalose dyring: A novel replacement of freeze-drying" BioPharm. (1991) 4:47-53.
Colaco et al., "Extraordinary stability of enzymes dried in trehalose: Simplified molecular biology" BioTech. (1992) 10:1007-1011.
Roser et al., "A sweeter way to fresher food" New Scientist (May 1993) pp. 25-28.
Madzarovova-Nohejlova, "Trehalase deficiency in a family" Gastroenterol. (1973) 65:130-133.
Blair Julian
Roser Bruce J.
Howard Sharon
Lehnhardt Susan K.
Page Thurman K.
Quadrant Holdings Cambridge Ltd.
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