Radionuclide labeling of vitamin B.sub.12 and coenzymes thereof

Details Radionuclide labeling of vitamin B.sub.12 and coenzymes thereof Radionuclide labeling of vitamin B.sub.12 and coenzymes thereof

1995-11-13

1998-04-14

Gitomer, Ralph

Organic compounds -- part of the class 532-570 series

Organic compounds

Carbohydrates or derivatives

536 264, 424 9, A61K 4900, C07H 2300

Patent

active

057393133

ABSTRACT:
A compound useful for in vivo imaging of organs and tumors is provided of formula: ##STR1## wherein ##STR2## is a cobalamin, ##STR3## is derived from a corrin carboxylic acid group of said cobalamin, Y is a linking group and X is a chelating group, optionally comprising a detectable radionuclide or a paramagnetic metal ion, and n is 1-3.

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