Radiolabeled N-substituted-6-iodo-3,14-dihydroxy-4,5.alpha.-epox

Details Radiolabeled N-substituted-6-iodo-3,14-dihydroxy-4,5.alpha.-epox Radiolabeled N-substituted-6-iodo-3,14-dihydroxy-4,5.alpha.-epox

1991-06-14

1993-05-04

Stoll, Robert L.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

424 11, 424 9, A61K 4300, A61K 4902, C07D48908

Patent

active

052083381

ABSTRACT:
The present invention is directed to radiolabeled N-substituted-6-iodo-3,14-dihydroxy-4,5.alpha.-epoxymorphinans, intermediates for producing the same, and a process for the preparation and methods of detecting opioid receptors.
The radioimaging agent of the present invention has the following formula: ##STR1## wherein I is selected from the group consisting of .sup.123 I and .sup.125 I; and where R is alkyl, cycloalkylloweralkyl or allyl.

REFERENCES:
patent: 4064228 (1977-12-01), Gross
patent: 4241065 (1980-12-01), Boswell, Jr. et al.
patent: 4451470 (1984-05-01), Ganti
patent: 4678779 (1987-07-01), Meyers et al.
patent: 4767718 (1988-08-01), Meyers
patent: 4775759 (1988-10-01), Rice et al.

Affiliated with

Also associated with

Rating

Radiolabeled N-substituted-6-iodo-3,14-dihydroxy-4,5.alpha.-epox does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Radiolabeled N-substituted-6-iodo-3,14-dihydroxy-4,5.alpha.-epox, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Radiolabeled N-substituted-6-iodo-3,14-dihydroxy-4,5.alpha.-epox will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-1976117