Radioiodinated dopamine receptor ligand

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

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252645, 424 11, 424 9, 436504, C07D47110, C09K 1104, G01N 33567

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active

046562800

ABSTRACT:
A process for the production of radioiodinated spiperone and certain derivatives thereof, and novel compositions made by the process. The process includes reacting spiperone, thallium trichloride and radioiodine in a sealed reaction vial. The novel compounds are useful for diagnosis of disease states resulting in quantitative changes in dopaminergic receptors.

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