Pyrrolylaminopiperidines

Details Pyrrolylaminopiperidines Pyrrolylaminopiperidines

1983-09-19

1984-06-05

Bond, Robert T.

Drug, bio-affecting and body treating compositions

Antigen, epitope, or other immunospecific immunoeffector

Parasitic organism or component thereof or substance...

546208, A61K 37445, C07D40312, C07D40304

Patent

active

044528035

ABSTRACT:
This invention relates to pyrrolylaminopiperidines and related compounds of the formula ##STR1## where R is hydrogen, loweralkyl, Arloweralkyl, cycloalkylloweralkyl, loweralkenyl and thienylloweralkyl; R.sub.1 is lower alkyl, hydrogen, loweralkylcarbonyl, loweralkoxycarbonyl, loweralkylthiocarbonyl of the formula ##STR2## cyano, loweralkylaminocarbonyl, diloweralkylaminocarbonyl, cycloalkylcarbonyl, cycloalkylloweralkylcarbonyl and loweralkenylcarbonyl; R.sub.2 is hydrogen, halogen and methyl; and the pharmaceutically acceptable acid addition salts thereof.

REFERENCES:
patent: 4348524 (1982-09-01), Karrer et al.
Flitsch et al., "Chem. Ber." vol. 102, pp. 3268-3276 (1969).
Scheibye et al., "Bull. Soc. Chim. Belg." vol. 87, No.(3), pp. 22 & 238 (1978).
Epton, "Chemistry and Industry", pp. 425-426 (Mar. 6, 1965).
Johnson et al. "J. Med. Chem.", vol. 24, pp. 1314-1319 (1961).
Neimegeers et. al., "Arzneim-Forsch.) (Drug. Res.) vol. 26, No. 8, pp. 1551-1556 (1976).
Janssen et al. "Arzneim-Forsch.) vol. 13, pp. 502-507 (1963).

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