Pyrrolopyridine derivatives and their use as Crth2 antagonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C546S112000

Reexamination Certificate

active

07666878

ABSTRACT:
There are provided according to the invention compounds of formula (I),in free or salt form, wherein R1, R2, R3, R 4, R5, R6, Q, W, X, m, n and p are as described in the specification, process for preparing them, and their use as pharmaceuticals.

REFERENCES:
patent: 5212195 (1993-05-01), Clark et al.
patent: 6248753 (2001-06-01), Chen
patent: 2008/0287416 (2008-11-01), Sandham et al.
patent: 2008/0312229 (2008-12-01), Sandham et al.
patent: 2008/0312230 (2008-12-01), Sandham
patent: 1 424 325 (2004-06-01), None
patent: 1 505 061 (2005-02-01), None
patent: 9507910 (1995-03-01), None
patent: WO 95/07910 (1995-03-01), None
patent: WO 95/33748 (1995-12-01), None
patent: WO 02/34747 (2002-05-01), None
patent: WO 03/066047 (2003-08-01), None
patent: WO 2004/007451 (2004-01-01), None
patent: WO 2005/040112 (2005-05-01), None
patent: WO 2005/121141 (2005-12-01), None
Andrew Brodrick et al, “1H-Pyrrolo[2,3-b]pyridines. Part III. A Novel Synthetic Route From 1-Substituted 2-Aminopyrroles” J. Organic Chemistry 19:1910-1913, 1975.
Anthony Verbiscar, “Synthesis of 1-p-Chlorobenzy1-7-azaindole-3-alpha-piperidylmethanol as a Potential Antimalarial Agent” J. Medicinal Chemistry 15(2):149-152, 1975.
Adberrahim Mouaddib et al., “Synthesis of Indolo[3,2-c]quinoline and Pyrido[3',2':4,5][3,2-c]quinoline Derivatives” Synthesis 4:549-556, 2000.
Adberrahim Mouaddib et al., “Synthesis of Benzo[5'6']cyclohepta[4,5] pyrrolo[2,3-beta]pyridin-12-one” Tetrahedron Letters 40:5853-5854, 1999.
C. Nicholas Hodge et al., “Corticotropin-Releasing Hormone Receptor Antagontists: Framework Design and Synthesis Guided . . . ” J. Med. Chem. 42:819-832, 1999.
Yakhontov et al., Khimiya Geterotsiklicheskikh Soedinenii 1:141-144, 1967.
Yakhonotov et al., Biol. Aktivn. Soedin, Akad. Nauk SSSR pp. 83-90, 1965.

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