Pyrazolopyrimidines as CRF antagonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C544S281000

Reexamination Certificate

active

06958341

ABSTRACT:
The present invention relates to pyrazolopyrimidines according to formula (I)and stereoisomers, isomers and salts thereof wherein R1-R5are selected from certain alkyl, aryl and heteroaryl species as defined in the specification wherein all of the compounds are useful as CRF antagonists and are thus useful in the treatment of neurological disorders as well as a multitude of other CRF associated diseases or conditions.

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