Pyrazolo benzodiazepines

Details Pyrazolo benzodiazepines Pyrazolo benzodiazepines

1977-03-07

1978-12-19

Trousof, Natalie

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

548374, 548378, 548373, 2602393T, 424273P, C07D48704

Patent

active

041307160

ABSTRACT:
Compounds are presented of the formula ##STR1## wherein R.sub.1 is selected from the group consisting of hydrogen, amino, halogen and nitro; R.sub.2 is selected from the group consisting of hydrogen, lower alkyl, carboxylic acids, esters and primary, secondary or tertiary amides thereof, alkylhydroxy, acylhydroxy-lower alkyl, amino-lower alkyl, alkylamino-lower alkyl, acylamino-lower alkyl and carboxaldehyde; and X is hydrogen or halogen and the pharmaceutically acceptable salts thereof.
Also presented are processes to produce the above compounds and intermediates thereof. These compounds exhibit pharmacological activity as anxiolytics, sedatives, muscle relaxants and anticonvulsants.

REFERENCES:
patent: 3910946 (1975-10-01), Gall
patent: 3927016 (1975-12-01), Hester
Chem. Abs., 8th coll., 26385S.

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