Pyrazolo[4,3-c]quinoline-3-one and imidazo[4,3-c]cinnolin-3-one

Details Pyrazolo[4,3-c]quinoline-3-one and imidazo[4,3-c]cinnolin-3-one Pyrazolo[4,3-c]quinoline-3-one and imidazo[4,3-c]cinnolin-3-one

1985-11-05

1987-09-01

Ford, John M.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

514248, 546 82, 544234, A61K 31415, C07D47104, C07D23728

Patent

active

046909303

ABSTRACT:
Compounds of the formula (I): ##STR1## wherein R.sup.1 and R.sup.2 each is hydrogen, alkyl, alkoxycarbonyl, carboxy, halogen, nitro or trifluoromethyl, or R.sup.1 and R.sup.2 taken together may form alkylene; R.sup.3 is hydrogen, alkyl, alkanoyl or alkylsulfonyl; R.sup.4 is hydrogen, alkoxycarbonyl, carboxy or halogen; X is hydrogen, alkyl, alkoxy, halogen or hydroxy; and Y is methine or nitrogen or salts thereof are provided. The compounds (I) show potent psychotropic activity.

REFERENCES:
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