Pyrazole derivatives as GnRH inhibitors

Details Pyrazole derivatives as GnRH inhibitors Pyrazole derivatives as GnRH inhibitors

2007-08-07

2007-08-07

Stockton, Laura L. (Department: 1626)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C514S404000, C514S339000, C514S341000, C548S364100, C546S276100

Reexamination Certificate

active

10525111

ABSTRACT:
The invention relates to a group of novel thieno-pyrrole compounds of Formula (I):wherein: R1, R2, R5, R6, R6a, R7, R8, A, B and M are as defined in the specification, which are useful as gonadotrophin releasing hormone antagonists. The invention also relates to pharmaceutical formulations of said compounds, methods of treatment using said compounds and to processes for the preparation of said compounds.

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