Pyrazole derivative, drug composition containing the same...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Carbohydrate doai

Reexamination Certificate

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Details

C514S025000, C514S866000, C536S004100, C536S018100

Reexamination Certificate

active

07576064

ABSTRACT:
The present invention provides pyrazole derivatives represented by the general formula:wherein R1represents H, an optionally substituted C1-6alkyl, etc.; one of Q and T represents a group selected from the following:and the other represents -Z-Ar wherein Z represents —O—, —S—, etc.; Ar represents an optionally substituted C6-10aryl, etc.;R represents an optionally substituted C3-8cycloalkyl, an optionally substituted C6-10aryl, etc., pharmaceutically acceptable salts thereof, and prodrugs thereof, which exhibit an excellent inhibitory activity in human sodium/glucose cotransporter (SGLT) and are useful as agents for the prevention, inhibition of progression or treatment of a disease associated with the excess uptake of at least a kind of carbohydrates selected from glucose, fructose and mannose (diabetes, postprandial hyperglycemia, impaired glucose tolerance, diabetic complications, etc.), and pharmaceutical compositions containing the same, medicinal uses thereof and intermediates for production therefor.

REFERENCES:
patent: 4526895 (1985-07-01), Jarreau et al.
patent: 2002/0052326 (2002-05-01), Mathias et al.
patent: 2004/0006025 (2004-01-01), Ohsumi et al.
patent: 2004/0063646 (2004-04-01), Fujikura et al.
patent: 2004/0110936 (2004-06-01), Ohsumi et al.
patent: 2004/0116357 (2004-06-01), Fushimi et al.
patent: 2004/0176308 (2004-09-01), Shiohara et al.
patent: 1568380 (2005-08-01), None
patent: WO 02/088157 (2002-11-01), None
patent: WO 02/098893 (2002-12-01), None
patent: WO2004/050122 (2004-06-01), None

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