Pyrazole analogs acting on cannabinoid receptors

Details Pyrazole analogs acting on cannabinoid receptors Pyrazole analogs acting on cannabinoid receptors

2008-07-01

2008-07-01

Saeed, Kamal A (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

C514S217080, C514S326000, C514S406000, C540S603000, C546S211000, C548S364100

Reexamination Certificate

active

10790498

ABSTRACT:
One aspect of the invention is concerned with cannabimimetic pyrazole analogs. Another aspect of the invention is concerned with new and improved pyrazole analogs having high affinities and/or selectivities for the CB1 cannabinoid receptor. A further aspect of the invention is concerned with pharmaceutical preparations employing the inventive analogs and methods of administering therapeutically effective amounts of the inventive analogs to provide a physiological effect.

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