Pyrazol-1-yl benzodiazepines and oximes thereof

Details Pyrazol-1-yl benzodiazepines and oximes thereof Pyrazol-1-yl benzodiazepines and oximes thereof

1978-09-14

1979-05-08

Ford, John M.

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C07D23114

Patent

active

041537998

ABSTRACT:
Compounds are presented of the formula ##STR1## wherein R.sub.1 is selected from the group consisting of hydrogen, amino, halogen and nitro; R.sub.2 is selected from the group consisting of hydrogen, lower alkyl, carboxylic acids, esters and primary, secondary or tertiary amides thereof, alkylhydroxy, acylhydroxy-lower alkyl, amino-lower alkyl, alkylamino-lower alkyl, acylamino-lower alkyl and carboxaldehyde; and X is hydrogen or halogen and the pharmaceutically acceptable salts thereof.
Also presented are processes to produce the above compounds and intermediates thereof. These compounds exhibit pharmacological activity as anxiolytics, sedatives, muscle relaxants and anticonvulsants.

REFERENCES:
patent: 3929766 (1975-12-01), Metlesics
patent: 4022800 (1977-05-01), Gschwend
patent: 4099012 (1978-07-01), Gschwend
Heckendorn et al., Chem. Abst. 1976, vol. 84, No. 121844w.
Allgeier et al., Chem. Abst. 1976, vol. 84, No. 180231s.

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