Pyrazinoic acid esters as antituberculosis agents

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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514924, 544406, A61K 31495, C07D24114, C07D24116, C07D24118

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active

049621114

ABSTRACT:
Pyrazinoic esters have been prepared. Compounds of this group are effective against mycobacteria including Mycobacteria tuberculosis, pyrazinamide-resistant Mycobacteria tuberculosis, Mycobacteria bovis and Mycobacteria kansasii.

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Suzuki, M., et al., Takamine Kenyusho Nempo 10:19-23 (1958), The Annual Report of Takamine Laboratory, vol. X.
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Ul'Yanova et al, Chem. Abst. 79-125379t (1973).

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