Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2005-06-01
2008-03-25
Saeed, Kamal A. (Department: 1626)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C514S359000, C514S575000, C564S123000
Reexamination Certificate
active
07348437
ABSTRACT:
Activity-based compositions for analyzing metalloproteases are disclosed, where the compositions include a chemical compound including a hydroxamate moiety and a benzophenone moiety. Methods for synthesizing these compounds are also disclosed, as well as methods of using them for determining the bioactivity of a compositions comprising active compounds toward a metalloproteases and for determining the potency of an inhibitor against a metalloprotease.
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Cravatt Benjamin F.
Jessani Nadim
Joseph Arul
Saghatelian Alan
Coppins Janet L.
DLA Piper (US) LLP
Saeed Kamal A.
The Scripps Research Institute
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