Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1997-11-07
2000-01-18
Shah, Mukund J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
514185, 540454, 540467, A01N 4300, A01N 5502, C07D26722
Patent
active
060158077
ABSTRACT:
This invention provides novel bis-indolylmaleimide macrocycle derivatives of the formula: and solvates thereof. The invention further provides the preparation, pharmaceutical formulations and the methods of use for inhibiting Protein Kinase C in mammals.
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Engel Gary Lowell
Farid Nagy Alphonse
Faul Margaret Mary
Jirousek Michael Robert
Richardson Lori Ann
Darkes Paul R.
Eli Lilly and Company
Shah Mukund J.
Truong Tamthom N.
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