Proline phosphonate derivatives

Details Proline phosphonate derivatives Proline phosphonate derivatives

1994-04-28

1996-08-06

Scheiner, Toni R.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Peptide containing doai

514 87, 514 89, 514 94, 548412, 548111, 546 21, 540542, 540450, 544 53, 544 57, 544 88, 544106, 558170, A61K 3800, A61K 3167, A01N 5700, C07F 502

Patent

active

055433960

ABSTRACT:
Peptidyl derivatives of diesters of .alpha.-aminoalkylphosphonic acids, particularly those with proline or related structures, their use in inhibiting serine proteases with chymotrypsin-like, trypsin-like, elastase-like, and dipeptidyl peptidase IV specificity and their roles as anti-inflammatory agents, anticoagulants, and anti-tumor agents.

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