Production of 2',3'-dideoxy-2',3'-didehydronucleosides

Details Production of 2',3'-dideoxy-2',3'-didehydronucleosides Production of 2',3'-dideoxy-2',3'-didehydronucleosides

1991-04-29

1992-07-14

Rollins, John W.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carbohydrates or derivatives

536 24, C07H 1700

Patent

active

051304210

ABSTRACT:
There are disclosed novel processes for producing 2',3'-dideoxy-2'3'-didehydronucleosides, for example, 2',3'-dideoxy-2',3'-didehydrothymidine in high yields and on a large scale. The compounds so-produced are useful as antiviral agents, especially as agents effective against the human immunodeficiency viruses (HIV).

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