Prodrugs of proton pump inhibitors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C546S273700

Reexamination Certificate

active

06897227

ABSTRACT:
Prodrugs of proton pump inhibitors of Formulas 1 through 4,where the symbols are as defined in the specification, and the R group includes at least one acidic group or its pharmaceutically acceptable salt, have improved aqueous solubility and bioavailability.

REFERENCES:
patent: 4045563 (1977-08-01), Berntsson et al.
patent: 4255431 (1981-03-01), Junggren et al.
patent: 4628098 (1986-12-01), Nohara et al.
patent: 4686230 (1987-08-01), Rainer et al.
patent: 4758597 (1988-07-01), Martin et al.
patent: 4965269 (1990-10-01), Brandstrom et al.
patent: 5021433 (1991-06-01), Alminger et al.
patent: 5045522 (1991-09-01), Kidd
patent: 5430042 (1995-07-01), Lindberg et al.
patent: 5693818 (1997-12-01), Von Unge
patent: 5708017 (1998-01-01), Dave et al.
patent: 6093734 (2000-07-01), Garst et al.
patent: 6599167 (2003-07-01), Waltz
patent: WO 0009498 (2000-02-01), None
patent: WO 0200166 (2002-01-01), None
patent: WO 0230920 (2002-04-01), None
Bundgaard, H., Design of Prodrugs, 1985, chapter 1, Elsevier Science Publishers B.V., not available.
Bundgaard, et al., Int. J. of Pharmaceutics, 1984, 45-56, 22, Elsevier.
Bundgaard, et al., Int. J. of Pharmaceutics, 1986, 19-28, 29, Elsevier.
Bundgaard, et al., J. Med. Chem, 1989, 2503-2507, 32.
Bundgaard, et al., Chem. Abstracts, 1980, vol. 93, abst. # 137935y.
Bundgaard, et al., Chem. Abstracts, 1981, vol. 95, abst. # 138493f.
Bundgaard, et al. Chem. Abstracts, 1981, vol. 95, abst. # 138592n.
Alminger, et al., Chem. Abstracts, 1989, vol. 110, abst. # 57664p.
Buur, et al., Chem. Abstracts, 1991, vol. 115, abst. # 64029s.
Hansen, et al., Chem. Abstracts,1991, vol. 115, abst. # 189582y.
Bundgaard, et al., Chem. Abstract, 1992, vol. 117, abst. # 14347q.
Jensen, et al., Chem. Abstract, 1992, vol. 117, abst. # 55790x.
Thomsen et al., Chem. Abstract, 1995, vol. 123, abst. # 17593b.
Sih, et al., Journal of Medicinal Chemistry, 1991, 1049-1062, 34.

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