Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2006-04-25
2006-04-25
Rao, Deepak (Department: 1624)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S272000, C514S275000, C544S123000, C544S321000, C544S326000, C544S327000, C544S328000, C544S329000
Reexamination Certificate
active
07034019
ABSTRACT:
The present invention concerns compounds of formula (A1)(A2)N—R1(I),the N-oxide forms, the pharmaceutically acceptable addition salts, the quaternary amines and stereochemically isomeric forms thereof, wherein R1is substituted C1-6alkyl; —S(═O)—R8; —S(═O)2—R8; C7-12alkylcarbonyl; optionally substituted C1-6alkyloxycarbonylC1-6alkylcarbonyl; with R8being C1-6alkyl, aryl1or Het1; (A1)(A2)N— is the covalently bonded form of the corresponding intermediate of formula (A1)(A2)N—H, which is a HIV replication inhibiting pyrimidine of formula
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De Corte Bart Lieven Daniel
de Jonge Marc René
Heeres Jan
Janssen Paul Adriaan Jan
Kavash Robert William
Donnelly Laura
Janssen Pharmaceutica N.V.
Rao Deepak
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