Processes for the production of chinazoline alkaloids

Organic compounds -- part of the class 532-570 series – Organic compounds – Chalcogen in the nitrogen containing substituent

Reexamination Certificate

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C544S093000, C544S094000, C544S249000, C544S250000

Reexamination Certificate

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07495096

ABSTRACT:
Processes for the production of a compound of the following formula (I)by converting a compound of formula (II) with 2-pyrrolidone used in excess relative to compound (II) and processes for the production of a compound of formula (III).The latter process includes preparing compound (I); a reduction reaction which yields compound (III) in salt form; and liberating compound (III) from the salt.

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