Processes for preparing polymorphic forms of...

Details Processes for preparing polymorphic forms of... Processes for preparing polymorphic forms of...

2008-12-15

2011-11-15

Chang, Celia (Department: 1625)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C514S230500

Reexamination Certificate

active

08058443

ABSTRACT:
Polymorphic forms of 3-(4-amino-1-oxo-1,3 dihydro-isoindol-2-yl)-piperidine-2,6-dione are disclosed. Compositions comprising the polymorphic forms, methods of making the polymorphic forms and methods of their use are also disclosed.

REFERENCES:
patent: 3536809 (1970-10-01), Applezweig
patent: 3598123 (1971-08-01), Zaffaroni et al.
patent: 3845770 (1974-11-01), Theeuwes et al.
patent: 3916899 (1975-11-01), Theeuwes et al.
patent: 4008719 (1977-02-01), Theeuwes et al.
patent: 4810643 (1989-03-01), Souza
patent: 4999291 (1991-03-01), Souza
patent: 5059595 (1991-10-01), Le Grazie
patent: 5073543 (1991-12-01), Marshall et al.
patent: 5120548 (1992-06-01), McClelland et al.
patent: 5229496 (1993-07-01), Deeley et al.
patent: 5354556 (1994-10-01), Sparks et al.
patent: 5385901 (1995-01-01), Kaplan et al.
patent: 5391485 (1995-02-01), Deeley et al.
patent: 5393870 (1995-02-01), Deeley et al.
patent: 5528823 (1996-06-01), Rudy, Jr. et al.
patent: 5580755 (1996-12-01), Souza
patent: 5591767 (1997-01-01), Mohr et al.
patent: 5593990 (1997-01-01), D'Amato
patent: 5629327 (1997-05-01), D'Amato
patent: 5635517 (1997-06-01), Muller et al.
patent: 5639476 (1997-06-01), Oshlack et al.
patent: 5674533 (1997-10-01), Santus et al.
patent: 5698579 (1997-12-01), Muller
patent: 5712291 (1998-01-01), D'Amato
patent: 5731325 (1998-03-01), Andrulis, Jr. et al.
patent: 5733566 (1998-03-01), Lewis
patent: 5798368 (1998-08-01), Muller et al.
patent: 5874448 (1999-02-01), Muller et al.
patent: 5877200 (1999-03-01), Muller
patent: 5929117 (1999-07-01), Muller et al.
patent: 5955476 (1999-09-01), Muller et al.
patent: 6020358 (2000-02-01), Muller et al.
patent: 6071948 (2000-06-01), D'Amato
patent: 6114335 (2000-09-01), Buerger et al.
patent: 6114355 (2000-09-01), D'Amato
patent: 6140346 (2000-10-01), Andrulis, Jr. et al.
patent: 6235756 (2001-05-01), D'Amato
patent: 6281230 (2001-08-01), Muller et al.
patent: 6316471 (2001-11-01), Muller et al.
patent: 6326388 (2001-12-01), Man et al.
patent: 6335349 (2002-01-01), Muller et al.
patent: 6380239 (2002-04-01), Muller et al.
patent: 6395754 (2002-05-01), Muller et al.
patent: 6403613 (2002-06-01), Man et al.
patent: 6420414 (2002-07-01), D'Amato
patent: 6458810 (2002-10-01), Muller et al.
patent: 6469045 (2002-10-01), D'Amato
patent: 6476052 (2002-11-01), Muller et al.
patent: 6518298 (2003-02-01), Green et al.
patent: 6555554 (2003-04-01), Muller et al.
patent: 7112602 (2006-09-01), D'Amato et al.
patent: 7465800 (2008-12-01), Jaworsky et al.
patent: 7855217 (2010-12-01), Jaworsky et al.
patent: 2001/0018445 (2001-08-01), Huang et al.
patent: 2001/0056114 (2001-12-01), D'Amato
patent: 2002/0035090 (2002-03-01), Zeldis et al.
patent: 2002/0045643 (2002-04-01), Muller et al.
patent: 2002/0052398 (2002-05-01), D'Amato
patent: 2002/0054899 (2002-05-01), Zeldis
patent: 2002/0061923 (2002-05-01), D'Amato
patent: 2002/0128228 (2002-09-01), Hwu
patent: 2002/0161023 (2002-10-01), D'Amato
patent: 2002/0173658 (2002-11-01), Muller et al.
patent: 2002/0183360 (2002-12-01), Muller et al.
patent: 2003/0013739 (2003-01-01), Masferrer et al.
patent: 2003/0028028 (2003-02-01), Man et al.
patent: 2003/0045552 (2003-03-01), Robarge et al.
patent: 2003/0069428 (2003-04-01), Muller et al.
patent: 2003/0096841 (2003-05-01), Robarge et al.
patent: 2003/0139451 (2003-07-01), Shah et al.
patent: 2003/0144325 (2003-07-01), Muller et al.
patent: 2003/0181428 (2003-09-01), Green et al.
patent: 2003/0187024 (2003-10-01), D'Amato
patent: 2003/0191098 (2003-10-01), D'Amato
patent: 2003/0235909 (2003-12-01), Hariri et al.
patent: 2004/0029832 (2004-02-01), Zeldis
patent: 2004/0077685 (2004-04-01), Figg et al.
patent: 2004/0077686 (2004-04-01), Dannenberg et al.
patent: 2004/0087546 (2004-05-01), Zeldis
patent: 2004/0091455 (2004-05-01), Zeldis
patent: 2004/0122052 (2004-06-01), Muller et al.
patent: 2004/0220144 (2004-11-01), Zeldis
patent: 2004/0266809 (2004-12-01), Emanuel et al.
patent: 2005/0203142 (2005-09-01), Zeldis
patent: 2006/0052609 (2006-03-01), Muller et al.
patent: 2008/0064876 (2008-03-01), Muller et al.
patent: 2008/0132541 (2008-06-01), Zeldis et al.
patent: 2009/0062343 (2009-03-01), Jaworsky et al.
patent: 2009/0149449 (2009-06-01), Liu et al.
patent: 2009/0149499 (2009-06-01), Jaworsky et al.
patent: 2009/0149500 (2009-06-01), Jaworski et al.
patent: 2009/0176832 (2009-07-01), Jaworsky et al.
patent: 2011/0015228 (2011-01-01), Jaworsky et al.
patent: A-H10-53576 (1998-02-01), None
patent: A-2001-503384 (2001-03-01), None
patent: WO97/46526(A1) (1997-12-01), None
patent: WO 98/03502 (1998-01-01), None
patent: WO98/03502(A1) (1998-01-01), None
patent: WO 98/54170 (1998-12-01), None
patent: WO 01/70275 (2001-09-01), None
patent: WO 01/87307 (2001-11-01), None
patent: WO2002/26737(A1) (2002-04-01), None
patent: WO 02/059106 (2002-08-01), None
patent: WO 02/064083 (2002-08-01), None
patent: PCT/US03/11578 (2003-01-01), None
patent: WO 03097052 (2003-11-01), None
patent: WO 2004103274 (2004-12-01), None
patent: WO 2005023192 (2005-03-01), None
patent: WO 2006/028964 (2006-03-01), None
patent: WO 2007/136640 (2007-11-01), None
patent: WO 2009/111948 (2009-09-01), None
patent: WO 2009/114601 (2009-09-01), None
patent: WO 2010/054833 (2010-05-01), None
patent: WO 2010/056384 (2010-05-01), None
patent: WO 2010/061209 (2010-06-01), None
patent: WO 2010/100476 (2010-09-01), None
patent: WO 2010/129636 (2010-11-01), None
patent: WO 2011/027326 (2011-03-01), None
patent: WO 2011/033468 (2011-03-01), None
patent: WO 2011/034504 (2011-03-01), None
patent: WO 2011/050590 (2011-05-01), None
patent: WO 2011/050962 (2011-05-01), None
patent: WO 2011/061611 (2011-05-01), None
patent: WO 2011/064574 (2011-06-01), None
Bernstein et al., 1999, “Concomitant Polymorphs,”Angew. Chem. Int. Ed., 38, 3440-61.
Byrn et al., 1999, “The X-Ray Powder Diffraction Method,”inSolid-State Chemistry of Drugs, 59-67.
Grant, 1999, “Theory and Origin of Polymorphism,”inPolymorphism in Pharmaceutical Solids, 1-33.
Hilfiker et al., 2006, Polymorphism in the Pharmaceutical Industry, 1-19, 287-308.
Remington et al., 1985, “Preformulation,”inRemington's Pharmaceutical Sciences, 1409-23.
Remington et al., 2000, “Preformulation,”inRemington: The Science and Practice of Pharmacy, 700-720.
Remington, 2006, Remington: The Science and Practice of Pharmacy, 21sted., 659-61.
Notice of Allowability mailed Oct. 13, 2010 in U.S. Appl. No. 12/335,395.
Office Action mailed Sep. 29, 2010 in U.S. Appl. No. 10/557,302.
Notice of Allowability mailed Mar. 23, 2011 in U.S. Appl. No. 12/220,336.
Threlfall, 2000, “Crystallisation of Polymorphs: Thermodynamic Insight into the Role of Solvent,”Organic Process Research&Development, 4, 384-90.
Office Action dated Apr. 16, 2010 in corresponding Japanese Patent Application No. 2006-525471 (with summary).
USPTO Office Action dated Oct. 10, 2007 in U.S. Patent 7,465,800.
Examiner Interview Summary mailed Mar. 7, 2011 in U.S. Appl. No. 12/220,336.
U.S. Appl. No. 60/499,723, filed Sep. 4, 2003, Jaworsky.
U.S. Appl. No. 60/372,348, filed Apr. 12, 2002, Hariri et al.
U.S. Appl. No. 09/545,654, filed Apr. 10, 2000, D'Amato.
U.S. Appl. No. 09/287,377, filed Apr. 7, 1999, D'Amato.
Bernstein, 2002, Polymorphism in Molecular Crystals, Clarendon Press, 115-18.
Bernstein, 2004, “Crystal Structure Prediction and Polymorphism,” ACA Transactions, 39, 14-23.
Bond et al., 2002, “Controlling Crystal Architecture in Molecular Solids: the Supramolecular Approach,”inSupramolecular Organization and Materials Design, Jones & Rao eds., Cambridge University Press, Chapter 12, pp. 391-443.
Brittain, 1999, “Methods for the Characterization of Polymorphs and Solvates,”inPolymorphism in Pharmaceutical Solids, Brittain ed., Chapter 6, pp. 227-278.
Brittain, 2002, “Polymorphism: Pharmaceutical Aspects,”inEncyclopedia of Pharmaceutical Technology, 2ndEdition, vol. 3, Swarbrick & Boylan eds., pp. 2239-2249.
Brittain, 2007, “Polymorphism and Solvatomorphism 2005,”

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