Processes for preparing anhydrous and hydrate forms of...

Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C514S317000

Reexamination Certificate

active

07135571

ABSTRACT:
The present invention is related to novel processes for preparing anhydrous and hydrated forms of piperidine derivatives, polymorphs and pseudomorphs thereof of the formulaswhich are useful as antihistamines, antiallergic agents and bronchodilators.

REFERENCES:
patent: 5204249 (1993-04-01), Schwartz
patent: 5375693 (1994-12-01), Woosley
patent: 5574045 (1996-11-01), Ortyl et al.
patent: 5578610 (1996-11-01), D'Ambra
patent: 5631375 (1997-05-01), King
patent: 5738872 (1998-04-01), Ortyl et al.
patent: 5855912 (1999-01-01), Ortyl et al.
patent: 5932247 (1999-08-01), Ortyl et al.
patent: 6037353 (2000-03-01), Woodward et al.
patent: 6039974 (2000-03-01), MacLaren et al.
patent: 6113942 (2000-09-01), Ortyl et al.
patent: 6147216 (2000-11-01), Krauss
patent: 6187791 (2001-02-01), Woodward et al.
patent: 6242606 (2001-06-01), Krauss
patent: 6399632 (2002-06-01), Woodward et al.
patent: 6613906 (2003-09-01), Davies et al.
patent: 1123438 (1982-05-01), None
patent: 1123439 (1982-05-01), None
patent: 2117892 (1993-10-01), None
patent: 2181089 (1994-12-01), None
patent: 117237 (2001-01-01), None
patent: 134917 (2001-07-01), None
patent: 134771 (2002-02-01), None
patent: WO 94/03170 (1994-02-01), None
patent: WO 94/09008 (1994-04-01), None
patent: WO 95/00480 (1995-01-01), None
patent: WO 96/26726 (1996-09-01), None
Bennett et al. “Concise chemical and technical dictionary” Chem. Pub. p. 553 (1976).
Evans et al. “An introduction to crystal chemistry” Cambridge p. 266-298, 396 (1964).
See copies in parent cases.
Rouli “The right stuff” Chem. Eng. News Feb. 24, p. 32-35 (2003).
Cheronis “semimicro experimental organic chemistry” De Graff p. 8, (1958).
Salole et al. “Effect of solvent deposition on . . . ” Derwent Acc. No. 86-22527 (1985).
Jalonen et al. “The crystal growth of carbamazepine . . . ” Derwent Acc. No. 90-02014 (1989).
Foks et al. “Effect of temperature and supersaturation . . . ” SciSearch 02857044 (1993).
Terao et al. “Second order nonliner . . . ” Pascal No. 92-0591460 (1990).
Internet page printout of Hawley's Condensed Chemical Dictionary 1 (14thed. 2002) (definitions of amorphous and conformation).
Chan, K.Y. et al.; Direct Enantiomerica Separation of Terfenadine and Its Major Acid Metabolite by High-Performance Liquid Chromatography, and the Lack of Stereoselective Terfenadine Enantiomer Biotransformation in Man; CA 116:50726 (1992).
Henton, D. et al; Process for Preparing Anhydrous and Hydrate of Antihistaminic Piperidine Derivatives (Polymorphs and Pseudomorphs); CA-124:202030 (1996).
Morrison, R.T. & Boyd, R.N.; Organic Chemistry 75 (1973).
Office Action dated May 26, 2004, in copending U.S. Appl. No. 10/162,011.
Office Action dated May 4, 2004, in copending U.S. Appl. No. 10/214,262.
Office Action dated Oct. 22, 2004, in copending U.S. Appl. No. 10/386,812.
Office Action dated May 17, 2004, in copending U.S. Appl. No. 10/125,094.
Office Action dated Apr. 18, 2003 in copending U.S. Appl. No. 10/125,094.
Eagleson, M.; Concise Encyclopedia Chemistry 872-873 (1944).
Cheronis, N.D.; Semimicro Experimental Organic Chemistry, A Laboratory Manual 16-17 (J de Gratt 1958).
English-Language Translation of Sep. 21, 2005, Letter from Seligsohn Gabrielli Levit & Co. to Israeli Registrar of Patents.
English-Language Translation of Nov. 1, 2005, Letter from Israeli Patent Office to Seligsohn Gabrielli Levit & Co.
English-Language Translation of Statement of Claim, C.F. 1088/06 (Israel Patent No. 134,917).
English-Language Translation of Urgent Application For Interlocutory Remedies, C.F. 1088/06 (Israel Patent No. 134,917).
English-Language Translation of Statement of Claim, C.F. 1152/05 (Israel Patent Nos. 117,237 and 134,771).
English-Language Translation of Urgent Application For Interlocutory Remedies, C.F. 1152/05 (Israel Patent Nos. 117,237 and 134,771).
Declaration of Prof. Joel Bernstein.
Declaration David E. Bugay, Ph.D.
English-Language Translation of Respondent's Reply to Application for Grant of Interlocutory Remedies, C.F. 1088/06.
Expert Opinion of Prof. Anthony Michael Glazer.
Report and Declaration of Peter W. Stephens.
Report and Declaration of Dr. Clare Grey.
Report and Declaration of Marc D. Hollingsworth, Ph.D.
English-Language Translation of Affidavit of Prof. Abraham Rubinstein.
English-Language Translation of Affidavit of Dr. Shmuel Cohen.
English-Language Translation of Affidavit of Mike Netz.
English-Language Translation of Affidavit of Netanel Aharonov.
English-Language Translation of Affidavit of Hagit Saban.
Letter from Thomas Irving to Liad Whatstein regarding Motion No. 2731/06 in C.F. 1088/06, dated Mar. 29, 2006.
Declaration of David E. Bugay, Ph.D., dated Apr. 2, 2006, and Exhibits A-E.
Declaration of Prof. Joel Bernstein, dated Apr. 2, 2006.
Urgent Application For Interlocutory Remedies, C.F. 1088/06 (Israel Patent No. 134,917).
Statement of Claim, C.F. 1088/06 (Israel Patent No. 134,917).
Statement of Reply, C.F. 1088/06 (Israel Patent No. 134,917) and English-language translation.
Respondent's Reply to Application for Grant of Interlocutory Remedies and English-language translation.
Applicant's Reply to Respondent's Response to the Application for Interlocutory Remedies, C.F. 1088/06 (Israel Patent No. 134,917) and English-language translation.
Ulicky, L. et al.; Comprehensive Dictionary of Physical Chemistry 21 (Prentice Hall 1992).
Dean, J.A.; Analytical Chemistry Handbook 10.24 (McGraw Hill 1995).
European Search Report in European Application No. 01124314.4-2101, dated Dec. 20, 2001.
PCT International Search Report in Application No. PCT/US95/04942, dated Aug. 10, 1995.
Canadian Office Action in Application No. 2,189,007, dated Nov. 6, 1998.
Argentine Search Report in Application No. 332047, dated Sep. 13, 1999.
Norwegian Search Report in Application No. 1996 4859, dated Nov. 21, 2001.
Office Action dated Jun. 26, 2003, in co-pending U.S. Appl. No. 10/162,011.
Office Action dated Apr. 18, 2003, in co-pending U.S. Appl. No. 10/125,094.
Office Action dated Aug. 8, 2003, in co-pending U.S. Appl. No. 10/214,262.
Amon, U. et al.; Anti-allergic effects of H1-receptor antagonists on histamin-containing cells; 178(8) Dermatologische Monatsschrift 327-33 (1992).
Bailey, D.G. et al.; Effect of Grapefruit Juice and Naringin on Nisoldipine Pharmacokinetics; 54(6) Clinical Pharmacology & Therapeutics 589-94 (1993).
Bailey, D.G. et al.; Grapefruit Juice—Felodipine Interaction: Mechanism, Predictability, and Effect of Naringin; 53 Clinical Pharmacology & Therapeutics 637-42 (1993).
Bailey, D.G. et al.; Grapefruit Juice and Drugs: How Significant is the Interaction; 26(2) Clinical Pharmacokinetics 91-98 (1994).
Bailey, D.G. et al.; Grapefruit Juice—Felodipine Interaction: Reproducibility and Characterization with the Extended Release Drug Formulation; 40 Br. J. Clinical Pharmacology 135-40 (1995).
Baroody, F. et al.; The Effects of H1antihistamines on the Early Allergic Response; 63 Annals of Allergy 551-55 (1989).
Cantilena, L. et al.; Effect of Cimetidine and Ranitidine on the Pharmacokinetics and ECG Pharmacodynamics of Terfenadine; 53(2) Clinical Pharmacology & Therapeutics 161 (1993).
Charlesworth, E.N. et al.; Cutaneous Late-Phase Response in Food-Allergic Children and Adolescents with Atopic Dermatitis; 23 Clinical and Experimental Allergy 391-98 (1993).
Crumb, W.J. et al.; Blockade of Multiple Human Cardiac Potassium Currents by the Antihistamine Terfenadine: Possible Mechanism for Terfenadine-Associated Cardiotoxicity; 47 Molecular Pharmacology 181-90 (1995).
Gupta, S.K. et al.; High-Performance Liquid Chromatographic Determination of Terfenadine in Commercial Tablets; 361 J. Chromatography 403-06 (1986).
Honig, P.K. et al.; Changes in the Pharmacokinetics and Electrocardiographic Pharmacodynamics of Terfenadine with Concomitant Administration of Erythromycin; 52(3) Clinical Pharmacology & Therapeutics 231-38 (1992).
Honig, P.K. et al.; Effect of Concomitant Administration of Cimetidine and

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